STRUCTURI GHID NAFTALENDIONICE INHIBITOARE ALE ADN TOPOIZOMERAZEI II LANŢ ALPHA

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Publication info:

No.: RO128627

Date: 30.07.2013

Inventor(s):

TAMAIAN RADU [RO]

NICULESCU VIOLETA-CAROLINA [RO]

ANGHEL NICOLAE-MIHAI [RO]

Applicant(s):
INST NAT CERCETARE DEZVOLTARE [RO]
Classification:
International patent classification (IPC):
C07D491/12; C07D491/22; G06F19/00

Cooperative patent classification (CPC):
Application info:
No.: RO20110000455
Date: 11.05.2011
Priority number(s):
RO20110000455 11.05.2011
BOPI:
Description:

Prezenta invenţie se referă la o serie de structuri-ghid, noi derivaţi naftalendionici tiolaţi, ce conţin structuri Markush, cu efect inhibitor asupra ADN topoizomerazei II lanţ α (ADN topo2 α).